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One-Pot Diastereoselective Synthesis of Spiro [pyrimidine-5, 8?-thiazolo [5, 4-f] quinoline] triones and Diimidazo-pyrazinyl-bis (1, 3-dimethyl-2, 4, 6-trioxohexahydropyrimidine-5-ylium) dihydrate as Anticancer Agents
Parmar, Mehul P; Chaudhari, Hrushikesh S; Vala, Disha P; Macwan, Pradip M; Nogales, Joaquina; Sahoo, Subash C; Salunke, Deepak B; Banerjee, Sourav; Chandra Sekhar, Kondapalli Venkata Gowri; Khan, Adam N;
The Journal of Organic Chemistry, Year: 2026
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Discovery of triazole-tethered glycinate and propanoate derivatives bearing a thiolactone moiety as quorum sensing inhibitors of Pseudomonas aeruginosa: design, synthesis, biological evaluation, and biofilm inhibition
Chaitanya, Kosana Sai; Yu, Tsz Tin; Chaudhari, Hrushikesh; Orenkonday, Nidhi; Kuthe, Pranali Vijaykumar; Kumar, Naresh; Dey, Ruchi Jain; Murugesan, Sankaranarayanan; Gowri Chandra Sekhar, Kondapalli Venkata;
RSC advances, Year: 2026, Vol: 16, Pages: 27977-27993
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Nitro-thiochromene derivatives as promising anti-leishmanial agents: Synthesis, biological evaluation, and in silico insights
7. Jatin Malik, Estela Melcon-Fernandez, Rafael Balana Fouce, Chandra Sekhar Kondapalli Venkata Gowri, Murugesan Sankaranarayanan;
Journal of Molecular Structure, Year: 2026, Vol: 1356, Pages: 145170
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Design, Synthesis and Evaluation of Indole?Based 1, 2, 3?Triazoles as Potential Quorum Sensing and Biofilm Inhibitors Against Pseudomonas aeruginosa
Chaitanya, Kosana Sai; Yu, Tsz Tin; Chaudhari, Hrushikesh; Orekonday, Nidhi; Kumar, Naresh; Dey, Ruchi Jain; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Archiv der Pharmazie, Year: 2026, Vol: 359, Pages: e70209
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Targeted HDAC8 inhibition with non-hydroxamate [1, 2, 4] triazolo [4, 3-a] quinoline compounds
Bandaru, NVM Rao; Fathima, Ashna; Sengar, Suryansh; Schweipert, Markus; Chaitanya, Kosana Sai; Mohammed, Muzaffar-Ur-Rehman; Gore, Suraj T; Jamma, Trinath; Sharma, Vivek; Abbineni, Chandrasekhar;
Scientific Reports, Year: 2026, Vol: 16, Pages: 7472
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Spirochromanone Cst-17 as a potent microtubule destabilizing agent showing anticancer effects in HeLa cells by binding to tubulin
5. Ranita Roy, Adinarayana Nandikolla, Debabrata Ghosh Dastidar, Urmi Chatterji, Kondapalli Venkata Gowri Chandra Sekhar, and Gopal Chakrabarti;
Scientific Publication, Year: 2026
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2-(1H-Pyrazol-1-yl) pyrimidine derivatives as promising anticancer candidates: synthesis, biological studies, and computational insights
Talamadla, Mahesh Kumar; Moharir, Shreyash Rajendra; Katdare, Mihika; Sengar, Suryansh; Sharma, Vivek; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Journal of Molecular Structure, Year: 2025, Pages: 145158
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Recent advances in triazole hybrid molecules for the therapeutic management of neglected tropical diseases
Malik, Jatin; Karande, Gauri; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
RSC Medicinal Chemistry, Year: 2025, Vol: 16, Pages: 5292-5317
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Design, synthesis, and biological evaluation of (E)-3-amino-N?-substituted benzylidene-6-chloropyrazine-2-carbohydrazide derivatives as anti-mycobacterial agents
Kumar, Boddupalli Venkata Siva; Bhardwaj, Puja; Chaudhari, Hrushikesh S; Dey, Ruchi Jain; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic Chemistry, Year: 2025, Pages: 109206
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Zinc based organic metal complexes for OLED applications
Paul, J John; Chaitanya, Kosana Sai; Ganesan, R; Jha, Purushottam; Sekhar, Kondapalli Venkata Gowri Chandra; Sindhu, S;
Synthetic Metals, Year: 2025, Pages: 117980
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Harnessing SIRT1 activators for effective PCOS treatment: A new frontier
Moharir, Shreyash Rajendra; Talamadla, Mahesh Kumar; Bhardwaj, Puja; Banerjee, Arnab; Dey, Ruchi Jain; Sekhar, Kondapalli Venkata Gowri Chandra;
Biomedicine & Pharmacotherapy, Year: 2025, Vol: 190, Pages: 118361
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Eco-friendly polyethylene glycol (PEG-400): PEG mediated synthesis, in-vitro, molecular dynamics, DFT, docking, ADMET and MM-GBSA studies of novel sulfonamides as potential antioxidant agents
Santhosh, CR; Chinnam, Sampath; Chaudhari, Hrushikesh S; Sekhar, Kondapalli Venkata Gowri Chandra; Oduselu, Gbolahan O; Ahuja, Vishal; Chidambaram, Kumarappan; Kerru, Nagaraju; Madhu, GM;
Journal of Molecular Structure, Year: 2025, Vol: 1346, Pages: 143201
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Exploring the Anti?Tubercular Potential of 2?(1H?Pyrazol?1?yl) Pyrimidine: Design, Synthesis, Biological Evaluation and Molecular Docking Studies
Talamadla, Mahesh Kumar; Nandikolla, Adinarayana; Shobha, Singarapalle; Nayar, Pranav Pramod; Kumar, Muthyala Murali Krishna; Sankaranarayanan, Murugesan; Sekhar, Kondapalli Venkata Gowri Chandra;
Chemistry & Biodiversity, Year: 2025, Vol: 22, Pages: e202500321
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Exploration of quinoxaline triazoles as antimycobacterial agents: design, synthesis and biological evaluation
Kumar, Boddupalli Venkata Siva; Talamadla, Mahesh Kumar; Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Shetye, Gauri; Franzblau, Scott G; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic & Medicinal Chemistry Letters, Year: 2025, Vol: 121, Pages: 130177
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A critique review of fetal hemoglobin modulators through targeting epigenetic regulators for the treatment of sickle cell disease
Ala, Chandu; Ramalingam, Sivaprakash; Gowri, Chandra Sekhar Kondapalli Venkata; Sankaranarayanan, Murugesan;
Life Sciences, Year: 2025, Vol: 369, Pages: 123536
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Design, synthesis, and biological evaluation of substituted benzyl-triazolopyridine derivatives as non-hydroxamate based HDAC8 inhibitors
Bandaru, NVM Rao; Fathima, Ashna; Joshi, Vandana; Schweipert, Markus; Pathur, Obanna; Chaitanya, Kosana Sai; Jamma, Trinath; Sharma, Vivek; Abbineni, Chandrasekhar; Meyer-Almes, Franz-Josef;
European Journal of Medicinal Chemistry Reports, Year: 2025, Vol: 13, Pages: 100255
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Design and Synthesis of Novel Spiro [Chromane?2, 4??Piperidin]?4?One Derivatives: Anti?Proliferative Investigation and Molecular Docking Studies
Nakka, Srinuvasu; Sengar, Suryansh; Sai Chaitanya, Kosana; Swati; Chandu, Ala; Sankaranarayanan, Murugesan; Sharma, Vivek; Devunuri, Nagaraju; Gowri Chandra Sekhar, Kondapalli Venkata;
Asian Journal of Organic Chemistry, Year: 2025, Vol: 14, Pages: e202400604
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Exploring 4-morpholinopyrrolo-[2, 3-d]-pyrimidine derivatives as novel anti-cancer agents: Design, synthesis and biological studies
Nakka, Srinuvasu; Chaitanya, Kosana Sai; Sengar, Suryansh; Chandu, Ala; Sankaranarayanan, Murugesan; Sharma, Vivek; Devunuri, Nagaraju; Sekhar, Kondapalli Venkata Gowri Chandra;
Journal of Molecular Structure, Year: 2025, Vol: 1319, Pages: 139565
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Development and Biological Evaluation of Novel Spiro 4?Chromanones as Potent Quorum Sensing Inhibitors
Sai Chaitanya, Kosana; Gupta, Pooja; Chitti, Surendar; Khetmalis, Yogesh Mahadu; Chandu, Ala; Murugesan, Sankaranarayanan; Pasupuleti, Mukesh; Sekhar, Kondapalli Venkata Gowri Chandra;
Journal of Chemistry, Year: 2024, Vol: 2024, Pages: 8227205
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Design, synthesis, and anti-mycobacterial evaluation of 1, 8-naphthyridine-3-carbonitrile analogues
Khetmalis, Yogesh Mahadu; Shobha, Singarapalle; Nandikolla, Adinarayana; Chandu, Ala; Murugesan, Sankaranarayanan; Kumar, Muthyala Murali Krishna; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC advances, Year: 2024, Vol: 14, Pages: 22676-22689
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Recent developments in thiochromene chemistry
Murugappan, Solai; Kuthe, Pranali Vijaykumar; Sekhar, Kondapalli Venkata Gowri Chandra; Sankaranarayanan, Murugesan;
Organic & Biomolecular Chemistry, Year: 2024, Vol: 22, Pages: 6045-6079
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Design, synthesis and biological evaluation of novel pyrido-[2, 3-d]-pyrimidin-2-amine analogues as antimycobacterial agents
Kumar, Boddupalli Venkata Siva; Khetmalis, Yogesh Mahadu; Chaitanya, Kosana Sai; Chandu, Ala; Shetye, Gauri; Ma, Rui; Murugesan, Sankaranarayanan; Franzblau, Scott G; Sekhar, Kondapalli Venkata Gowri Chandra;
Journal of Molecular Structure, Year: 2024, Vol: 1303, Pages: 137600
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Tetrahydroisoquinoline based 5-nitro-2-furoic acid derivatives: a promising new approach for anti-tubercular agents
Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Sangeetha, Guruvelli Padma Vijaya; Chandu, Ala; Swati; Kumar, Muthyala Murali Krishna; Sharma, Vivek; Murugesan, Sankaranarayanan; Chandra Sekhar, Kondapalli Venkata Gowri;
New Journal of Chemistry, Year: 2023, Vol: 47, Pages: 15378-15389
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Design, synthesis, and biological evaluation of novel quinazolin-4 (3H)-one-based histone deacetylase 6 (HDAC6) inhibitors for anticancer activity
Khetmalis, Yogesh Mahadu; Fathima, Ashna; Schweipert, Markus; Debarnot, C?cile; Bandaru, Naga Venkata Madhusudhan Rao; Murugesan, Sankaranarayanan; Jamma, Trinath; Meyer-Almes, Franz-Josef; Sekhar, Kondapalli Venkata Gowri Chandra;
International Journal of Molecular Sciences, Year: 2023, Vol: 24, Pages: 11044
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Design, synthesis and biological evaluation of phenanthridine amide and 1, 2, 3-triazole analogues against Mycobacterium tuberculosis
Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Venkata Siva Kumar, Boddupalli; Chandu, Ala; Karan Kumar, Banoth; Shetye, Gauri; Ma, Rui; Murugesan, Sankaranarayanan; Franzblau, Scott G; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC Medicinal Chemistry, Year: 2023, Vol: 14, Pages: 1549-1561
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Molecular-level strategic goals and repressors in Leishmaniasis?Integrated data to accelerate target-based heterocyclic scaffolds
Abirami, M; Kumar, Banoth Karan; Dey, Sanchita; Johri, Samridhi; Reguera, Rosa M; Bala?a-Fouce, Rafael; Sekhar, Kondapalli Venkata Gowri Chandra; Sankaranarayanan, Murugesan;
European Journal of Medicinal Chemistry, Year: 2023, Vol: 257, Pages: 115471
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Visible light sensing of ions by a cyanoquinoxaline 1, 4-dioxide-based probe and its applications
Savita; Nandikolla, Adinarayana; Shukla, Adarash Kumar; Chandra Sekhar, Kondapalli Venkata Gowri; Bhattacharya, Anupam;
Dalton Transactions, Year: 2023, Vol: 52, Pages: 4103-4111
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Retrospective review of chromane analogues as anti-protozoal leads: a decade's worth of evolution
Jadhav, Snehal R; Karan Kumar, Banoth; Joshi, Renuka Parshuram; Suryakant, Chougule Kishor; Chandu, Ala; Muzaffar-Ur-Rehman, Mohammed; Khetmalis, Yogesh Mahadu; Nandikolla, Adinarayana; Murugesan, Sankaranarayan; Chandra Sekhar, Kondapalli VG;
Current Topics in Medicinal Chemistry, Year: 2023, Vol: 23, Pages: 713-735
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Design, synthesis, and antimycobacterial evaluation of novel tetrahydroisoquinoline hydrazide analogs
Kumar, Boddupalli Venkata Siva; Khetmalis, Yogesh Mahadu; Nandikolla, Adinarayana; Kumar, Banoth Karan; Van Calster, Kevin; Murugesan, Sankaranarayanan; Cappoen, Davie; Sekhar, Kondapalli Venkata Gowri Chandra;
Chemistry & Biodiversity, Year: 2023, Vol: 20, Pages: e202200939
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Design, synthesis, and biological evaluation of tetrahydroisoquinoline based hydroxamate derivatives as HDAC 6 inhibitors for cancer therapy
Khetmalis, Yogesh Mahadu; Shree, Bakhya; Kumar, Boddupalli Venkata Siva; Schweipert, Markus; Debarnot, C?cile; Ashna, Fathima; Sankaranarayanan, Murugesan; Trinath, Jamma; Sharma, Vivek; Meyer-Almes, Franz-Josef;
Journal of Molecular Structure, Year: 2023, Vol: 1278, Pages: 134952
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Inspection of in-house designed novel thiochromone amino-acid conjugate derivatives as Lm-NMT inhibitor?An in-silico analysis
Johri, Samridhi; Kumar, Banoth Karan; Dey, Sanchita; Balana-Fouce, Rafael; Sekhar, Kondapalli Venkata Gowri Chandra; Kunjiappan, Selvaraj; Murugesan, Sankaranarayanan;
Journal of Molecular Graphics and Modelling, Year: 2023, Vol: 119, Pages: 108397
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Design, Synthesis and Biological Evaluation of Novel Spiro?[Chroman?2, 4??Piperidin]?4?One Analogs as Anti?Tubercular Agents
Chitti, Surendar; Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Van Calster, Kevin; Kumar, Boddupalli Venkata Siva; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Cappoen, Davie; Sekhar, Kondapalli Venkata Gowri Chandra;
Chemistry & Biodiversity, Year: 2022, Vol: 19, Pages: e202200304
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Design, synthesis and biological evaluation of benzo-[d]-imidazo-[2, 1-b]-thiazole and imidazo-[2, 1-b]-thiazole carboxamide triazole derivatives as antimycobacterial agents
Chitti, Surendar; Van Calster, Kevin; Cappoen, Davie; Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Cos, Paul; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
RSC advances, Year: 2022, Vol: 12, Pages: 22385-22401
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Design, Synthesis and Anti-mycobacterial Evaluation of Imidazo-[1,2-a]-pyridine Analogues
Yogesh, M, K., Surendar, C., Anjani, U. W., Karan Kumar, B., Murali Krishna Kumar M., Murugesan, S., Chandra Sekhar, K.V.G;
RSC Medicinal Chemistry, Year: 2022, Vol: 13, Pages: 327-342
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Discovery of potent antitubercular agents: Design, synthesis and biological evaluation of 4-(3-(4-substitutedpiperazin-1-yl)-quinoxalin-2-yl)-naphthalen-1-ol analogues
Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Naidu, Kalaga Mahalakshmi; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Toxicology in Vitro, Year: 2022, Vol: 82, Pages: 105370
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Search for structurally diverse heterocyclic analogs as dual-acting antimalarial and antileishmanial agents: An overview
Dey, Sanchita; Johri, Samridhi; Abirami, M; Kumar, Banoth Karan; Taramelli, Donatella; Basilico, Nicoletta; Balana-Fouce, Rafael; Sekhar, Kondapalli Venkata Gowri Chandra; Murugesan, Sankaranarayanan;
European Journal of Medicinal Chemistry Reports, Year: 2022, Vol: 4, Pages: 100031
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Design, synthesis and evaluation of novel ?-carboline ester analogues as potential anti-leishmanial agents
Karan Kumar, Banoth; Faheem; Balana Fouce, Rafael; Melcon-Fernandez, Estela; Perez-Pertejo Yolanda, Yolanda; Reguera, Rosa M; Adinarayana, Nandikolla; Chandra Sekhar, Kondapalli Venkata Gowri; Vanaparthi, Satheeshvarma; Murugesan, Sankaranarayan;
Journal of Biomolecular Structure and Dynamics, Year: 2022, Vol: 40, Pages: 12592-12607
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Liquid chromatography-mass spectrometric methods for trace quantification of potential genotoxic impurities in ivacaftor and lumacaftor
Panchakarla, RK; Ravi, PR; Mullangi, S; Kondapalli, VGCS;
Annales Pharmaceutiques Fran?aises, Year: 2022, Vol: 80, Pages: 448-459
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Design, synthesis, and biological evaluation of phenyl thiazole-based AR-V7 degraders
Bhumireddy, Archana; Bandaru, NVM Rao; Reddy, B Raghurami; Gore, Suraj T; Mukherjee, Subhendu; Balasubramanian, Wesley Roy; Kumar, V Sumanth; Alapati, Krishna Satya; Sekhar, Kondapalli Venkata Gowri Chandra; Nellore, Kavitha;
Bioorganic & Medicinal Chemistry Letters, Year: 2022, Vol: 55, Pages: 128448
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Anti-infective potential of manzamine alkaloids-a review
Ashok, Penta; Kumar, Banoth K; Chander, Subhash; Chandra, Sekhar; Kondapalli, VG; Sankaranarayanan, Murugesan;
Medicinal Chemistry, Year: 2022, Vol: 18, Pages: 629-654
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Pharmacophore based virtual screening, molecular docking, molecular dynamics and MM-GBSA approach for identification of prospective SARS-CoV-2 inhibitor from natural product databases
Kumar, Banoth Karan; Faheem, n; Sekhar, Kondapalli Venkata Gowri Chandra; Ojha, Rupal; Prajapati, Vijay Kumar; Pai, Aravinda; Murugesan, Sankaranarayanan;
Journal of Biomolecular Structure and Dynamics, Year: 2022, Vol: 40, Pages: 1363-1386
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Medicinal chemistry perspectives of 1, 2, 3, 4-tetrahydroisoquinoline analogs?biological activities and SAR studies
Karan Kumar, Banoth; Sekhar, Chandra; Gowri, Kondapalli Venkata; Chander, Subhash; Kunjiappan, Selvaraj; Murugesan, Sankaranarayanan;
RSC advances, Year: 2021, Vol: 11, Pages: 12254-12287
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Selective and Sensitive UHPLC Method for the Trace Analysis of Formaldehyde in Drug Substance Using Fused-core Column Technology and Detailed Pre-column Derivatization study
Panchakarla, Ravi K; Ravi, Punna Rao; Chandra Sekhar, Kondapalli VG;
Current Pharmaceutical Analysis, Year: 2021, Vol: 17, Pages: 201-209
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Design, synthesis and evaluation of novel ?-carboline ester analogues as potential anti-leishmanial agents.
Banoth Karan Kumar, Faheem, Rafael Balana Fouce, Estela Melcon-Fernandez, Nandikolla Adinarayana, Kondapalli Venkata Gowri Chandra Sekhar, Satheeshvarma Vanaparthi & Sankaranarayan Murugesan;
Journal of Biomolecular Structure and Dynamics, Year: 2021, Pages: DOI: 10.1080/07391102.2021.1973564.
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1,2,3,4-Tetrahydroisoquinoline (THIQ) as privileged scaffold for anticancer de novo drug design.
Faheem, Banoth Karan Kumar, Kondapalli Venkata Gowri Chandra Sekhar, Subhash Chander, Selvaraj Kunjiappan & Sankaranarayanan Murugesan;
Expert Opinion on Drug Discovery, Year: 2021, Vol: 16, Pages: 1119-114
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Liquid chromatography?tandem mass spectrometric method for trace quantification of ethyl methanesulfonate: a genotoxic impurity in dapoxetine hydrochloride
Ravi Kiran Panchakarla, Punna Rao Ravi, Kondapalli Venkata Gowri Chandra Sekhar;
Future Journal of Pharmaceutical Sciences, Year: 2021, Vol: 7, Pages: 91
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1,8-naphthyridine derivatives: an updated review on recent advancements of their myriad biological activities.
Shivani Mithula, Adinarayana Nandikolla, Sankaranarayanan Murugesan & Venkata GCS Kondapalli;
Future Medicinal Chemistry, Year: 2021, Vol: 13, Pages: 1591-1618
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Novel phenanthridine amide analogs as potential anti-leishmanial agents: In vitro and in silico insights
Nandikolla, Adinarayana; Srinivasarao, Singireddi; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Aggarwal, Himanshu; Balana-Fouce, Rafael; Melc?n-Fernandez, Estela; P?rez-Pertejo, Yolanda; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic Chemistry, Year: 2021, Vol: 117, Pages: 105414
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Oxindole and its derivatives: A review on recent progress in biological activities
Khetmalis, Yogesh Mahadu; Shivani, Mithula; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Biomedicine & Pharmacotherapy, Year: 2021, Vol: 141, Pages: 111842
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Design, synthesis and biological evaluation of 7?(5?((substituted?amino)-methyl)-thiophen?2?yl)-spiro-[chroman?2, 4??piperidin]?4?one hydrochloride analogues as anticancer agents
Chitti, Surendar; Pulya, Sravani; Nandikolla, Adinarayana; Patel, Tarun Kumar; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Ghosh, Balaram; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic Chemistry, Year: 2021, Vol: 112, Pages: 104865
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Design, synthesis and biological evaluation of novel 1, 2, 3-triazole analogues of Imidazo-[1, 2-a]-pyridine-3-carboxamide against Mycobacterium tuberculosis
Nandikolla, Adinarayana; Srinivasarao, Singireddi; Khetmalis, Yogesh Mahadu; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Shetye, Gauri; Ma, Rui; Franzblau, Scott G; Sekhar, Kondapalli Venkata Gowri Chandra;
Toxicology in Vitro, Year: 2021, Vol: 74, Pages: 105137
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Recent Update on the Anti-infective Potential of ?-carboline Analogs
Faheem; Kumar, Banoth K; Sekhar, Kondapalli Venkata GC; Kunjiappan, Selvaraj; Jamalis, Joazaizulfazli; Balana-Fouce, Rafael; Sankaranarayanan, Murugesan;
Mini reviews in medicinal chemistry, Year: 2021, Vol: 21, Pages: 398-425
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Seeking potent anti-tubercular agents: design and synthesis of substituted-N-(6-(4-(pyrazine-2-carbonyl) piperazine/homopiperazine-1-yl) pyridin-3-yl) benzamide derivatives as anti-tubercular agents (vol 10, pg 12272, 2020)
Srinivasarao, Singireddi; Nandikolla, Adinarayana; Suresh, Amaroju; Van Calster, Kevin; De Vooght, Linda; Cappoen, Davie; Ghosh, Balaram; Aggarwal, Himanshu; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
RSC ADVANCES, Year: 2020, Vol: 10, Pages: 18907-18907
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Synthesis, study of antileishmanial and antitrypanosomal activity of imidazo pyridine fused triazole analogues
Nandikolla, Adinarayana; Srinivasarao, Singireddi; Karan Kumar, Banoth; Murugesan, Sankaranarayanan; Aggarwal, Himanshu; Major, Louise L; Smith, Terry K; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC advances, Year: 2020, Vol: 10, Pages: 38328-38343
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Inhibitors of pantothenate synthetase of Mycobacterium tuberculosis?a medicinal chemist perspective
Suresh, Amaroju; Srinivasarao, Singireddi; Khetmalis, Yogesh Mahadu; Nizalapur, Shashidhar; Sankaranarayanan, Murugesan; Sekhar, Kondapalli Venkata Gowri Chandra;
RSC advances, Year: 2020, Vol: 10, Pages: 37098-37115
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Druggable targets of SARS-CoV-2 and treatment opportunities for COVID-19
Kumar, Banoth Karan; Sekhar, Kondapalli Venkata Gowri Chandra; Kunjiappan, Selvaraj; Jamalis, Joazaizulfazli; Bala?a-Fouce, Rafael; Tekwani, Babu L; Sankaranarayanan, Murugesan;
Bioorganic chemistry, Year: 2020, Vol: 104, Pages: 104269
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Discovery of 1, 2, 3-triazole based quinoxaline-1, 4-di-N-oxide derivatives as potential anti-tubercular agents
Srinivasarao, Singireddi; Nandikolla, Adinarayana; Suresh, Amaroju; Ewa, Augustynowicz-Kopec; G?ogowska, Agnieszka; Ghosh, Balaram; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Pulya, Sravani; Aggarwal, Himanshu;
Bioorganic Chemistry, Year: 2020, Vol: 100, Pages: 103955
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Seeking potent anti-tubercular agents: design and synthesis of substituted-N-(6-(4-(pyrazine-2-carbonyl) piperazine/homopiperazine-1-yl) pyridin-3-yl) benzamide derivatives as anti-tubercular agents
Srinivasarao, Singireddi; Nandikolla, Adinarayana; Suresh, Amaroju; Calster, Kevin Van; De Voogt, Linda; Cappoen, Davie; Ghosh, Balaram; Aggarwal, Himanshu; Murugesan, Sankaranarayanan; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC advances, Year: 2020, Vol: 10, Pages: 12272-12288
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Visible-Light-Mediated Tandem Sulfonylation/Cyclization of Vinyl Azides with Sulfonyl Hydrazines for the Synthesis of 6-(Sulfonylmethyl) phenanthridines under Mild Conditions
Mao, Liu-Liang; Quan, Li-Xia; Zhu, Xian-Hong; Ji, Cong-Bin; Zhou, An-Xi; Chen, Fayun; Zheng, Da-Gui;
Synlett, Year: 2019, Vol: 30, Pages: 955-960
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Design, synthesis and biological evaluation of 1, 2, 3-triazole based 2-aminobenzimidazoles as novel inhibitors of LasR dependent quorum sensing in Pseudomonas aeruginosa
Srinivasarao, Singireddi; Nandikolla, Adinarayana; Nizalapur, Shashidhar; Yu, Tsz Tin; Pulya, Sravani; Ghosh, Balaram; Murugesan, Sankaranarayanan; Kumar, Naresh; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC advances, Year: 2019, Vol: 9, Pages: 29273-29292
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Design, synthesis and biological evaluation of 2-(3, 4-dimethoxyphenyl)-6 (1, 2, 3, 6-tetrahydropyridin-4-yl) imidazo [1, 2-a] pyridine analogues as antiproliferative agents
Chitti, Surendar; Singireddi, SrinivasaRao; Reddy, Pochana Santosh Kumar; Trivedi, Prakruti; Bobde, Yamini; Kumar, Chandan; Rangan, Krishnan; Ghosh, Balaram; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic & Medicinal Chemistry Letters, Year: 2019, Vol: 29, Pages: 2551-2558
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Design, synthesis and anti-tumour activity of new pyrimidine-pyrrole appended triazoles
Thiriveedhi, Arunkumar; Nadh, Ratnakaram Venkata; Srinivasu, Navuluri; Bobde, Yamini; Ghosh, Balaram; Sekhar, Kondapalli Venkata Gowri Chandra;
Toxicology in Vitro, Year: 2019, Vol: 60, Pages: 87-96
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Design, synthesis and biological evaluation of 5-(2-(4-(substituted benzo [d] isoxazol-3-yl) piperazin-1-yl) acetyl) indolin-2-one and 5-(2-(4-substitutedpiperazin-1-yl) acetyl) indolin-2-one analogues as novel anti-tubercular agents
Naidu, Kalaga Mahalakshmi; Gajanan, Rudresh Naik; Sekhar, Kondapalli Venkata Gowri Chandra;
Arabian Journal of Chemistry, Year: 2019, Vol: 12, Pages: 2418-2429
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Synthesis and activity of benzopiperidine, benzopyridine and phenyl piperazine based compounds against Leishmania infantum.
Subhash Chander, Subhash Chander; Penta Ashok, Penta Ashok; Reguera, RM; Perez-Pertejo, MY; Carbajo-Andres, R; Balana-Fouce, R; Sekhar, KVGC; Murugesan Sankaranarayanan, Murugesan Sankaranarayanan;
Scientific Publication, Year: 2018
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Experimental study of flow blurring twin fluid atomization concept using transparent injector
Murugan, R; Bollu, B; Sekhar, K; Kolhe, PS;
ICLASS 2018-14th International Conference on Liquid Atomization and Spray Systems, Year: 2018
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Sulfur?Assisted Deprotection of Methylene Nitrile Group: One?Pot Synthesis of 4?Substituted?2H?1, 2, 3?triazoles
Nagesh, Hunsur Nagendra; Singireddi, Srinivasarao; Suresh, Amaroju; Nizalapur, Shashidhar; Murugesan, Sankaranarayanan; Kanneboina, Kumar; Kumar, Naresh; Sekhar, Kondapalli Venkata Gowri Chandra;
ChemistrySelect, Year: 2018, Vol: 3, Pages: 7565-7571
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Synthesis and activity of benzopiperidine, benzopyridine and phenyl piperazine based compounds against Leishmania infantum
Chander, Subhash; Ashok, Penta; Reguera, Rosa M; Perez-Pertejo, M Yolanda; Carbajo-Andres, Ruben; Balana-Fouce, Rafael; Sekhar, Kondapalli Venkata Gowri Chandra; Sankaranarayanan, Murugesan;
Experimental parasitology, Year: 2018, Vol: 189, Pages: 49-60
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Design, Synthesis and Biological Evaluation of Triazole?Containing 2?Phenylindole and Salicylic Acid as Quorum Sensing Inhibitors Against Pseudomonas aeruginosa
Srinivasarao, Singireddi; Nizalapur, Shashidhar; Yu, Tsz Tin; Wenholz, Daniel Stanley; Trivedi, Prakruti; Ghosh, Balaram; Rangan, Krishnan; Kumar, Naresh; Gowri Chandra Sekhar, Kondapalli Venkata;
ChemistrySelect, Year: 2018, Vol: 3, Pages: 9170-9180
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Anti-proliferative activity, molecular modeling studies and interaction with calf thymus DNA of novel ciprofloxacin analogues: NARVA SURESH et al
Suresh, Narva; Suresh, Amaroju; Yerramsetty, Suresh; Bhadra, Manika Pal; Alvala, Mallika; Sekhar, Kondapalli Venkata Gowri Chandra;
Journal of Chemical Sciences, Year: 2018, Vol: 130, Pages: 121
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Design, synthesis of 9H-fluorenone based 1,2,3-triazole analogues as Mycobacterium tuberculosis InhA inhibitors
Suresh, A., Srinivasarao, S., Agnieszka, Ewa, Mallika, A., Lherbet, C, Chandra Sekhar, K.V.G.;
Chemical biology and drug design, Year: 2017, Vol: 91, Pages: 1078-1086
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Design and synthesis of 4-morpholino-6-(1, 2, 3, 6-tetrahydropyridin-4-yl)-N-(3, 4, 5-trimethoxyphenyl)-1, 3, 5-triazin-2-amine analogues as tubulin polymerization inhibitors
Narva, Suresh; Chitti, Surendar; Amaroju, Suresh; Bhattacharjee, Debanjan; Rao, Bala Bhaskara; Jain, Nishant; Alvala, Mallika; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic & Medicinal Chemistry Letters, Year: 2017, Vol: 27, Pages: 3794-3801
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Do spiroindolines have the potential to replace vesamicol as lead compound for the development of radioligands targeting the vesicular acetylcholine transporter?
Lindemann, Marcel; Deuther-Conrad, Winnie; Moldovan, Rares; Sekhar, Kondapalli Venkata Gowri Chandra; Brust, Peter; Wenzel, Barbara;
Bioorganic & Medicinal Chemistry, Year: 2017, Vol: 25, Pages: 5107-5113
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A Study on Socio Demographic Profile of Adult Female Smokers in Rural Areas of Srikakulam District, AP
Sravya, B; Susmitha, G; Chandra Sekhar, K; Mohan, Ch Rama; Deotale, PG;
Indian Journal of Public Health Research & Development, Year: 2016, Vol: 7
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Synthesis and biological evaluation of pyrrolo [2, 3-b] pyridine analogues as antiproliferative agents and their interaction with calf thymus DNA
Narva, Suresh; Chitti, Surendar; Bala, Bhaskara Rao; Alvala, Mallika; Jain, Nishant; Kondapalli, Venkata Gowri Chandra Sekhar;
European Journal of Medicinal Chemistry, Year: 2016, Vol: 114, Pages: 220-231
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Design, synthesis and biological evaluation of new substituted sulfonamide tetrazole derivatives as antitubercular agents
Suresh, Amaroju; Suresh, Narva; Misra, Sunil; Kumar, Muthyala Murali Krishna; Sekhar, Kondapalli Venkata Gowri Chandra;
ChemistrySelect, Year: 2016, Vol: 1, Pages: 1705-1710
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Multicomponent cascade reaction: dual role of copper in the synthesis of 1, 2, 3-triazole tethered benzimidazo [1, 2-a] quinoline and their photophysical studies
Nagesh, Hunsur Nagendra; Suresh, Amaroju; Reddy, Muthyala Nagarjuna; Suresh, Narva; Subbalakshmi, Jayanty; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC advances, Year: 2016, Vol: 6, Pages: 15884-15894
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Seeking potent anti-tubercular agents: Design, synthesis, anti-tubercular activity and docking study of various ((triazoles/indole)-piperazin-1-yl/1, 4-diazepan-1-yl) benzo [d] isoxazole derivatives
Naidu, Kalaga Mahalakshmi; Srinivasarao, Singireddi; Agnieszka, Napi?rkowska; Ewa, Augustynowicz-Kope?; Kumar, Muthyala Murali Krishna; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic & medicinal chemistry letters, Year: 2016, Vol: 26, Pages: 2245-2250
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Identification and development of pyrazolo [4, 3-c] pyridine carboxamides as Mycobacterium tuberculosis pantothenate synthetase inhibitors
Amaroju, Suresh; Kalaga, Mahalakshmi Naidu; Srinivasarao, Singireddi; Napi?rkowska, Agnieszka; Augustynowicz-Kope?, Ewa; Murugesan, Sankaranarayanan; Chander, Subhash; Krishnan, Rangan; Chandra Sekhar, Kondapalli Venkata Gowri;
New Journal of Chemistry, Year: 2016, Vol: 41, Pages: 347-357
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A Study of Nutritional Status of Adolescent Girls of Social Welfare Hostels in and around Vijayawada City.
Shridevi, K; Nageshwara Rao, R; Madhavi, P; Chandra Sekhar, K; Deotale, PG;
Indian Journal of Public Health Research & Development, Year: 2015, Vol: 6
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G, Biswas NN, Nizalapur S, Rice SA, Willcox M, Black DSt. C, Kumar N
Goh, WK; Gardner, CR; Chandra Sekhar, KV;
Bioorg. Med. Chem, Year: 2015, Vol: 23, Pages: 7366
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Synthesis and biological evaluation of novel phenanthridinyl piperazine triazoles via click chemistry as anti-proliferative agents
Nagesh, Hunsur Nagendra; Suresh, Narva; Prakash, Gollapalli Venkata Subrahmanya Bhanu; Gupta, Samarth; Rao, Janapala Venkateswara; Sekhar, Kondapalli Venkata Gowri Chandra;
Medicinal Chemistry Research, Year: 2015, Vol: 24, Pages: 523-532
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Novel amide and sulphonamide derivatives of 6-(piperazin-1-yl) phenanthridine as potent Mycobacterium tuberculosis H37Rv inhibitors
Naidu, Kalaga Mahalakshmi; Nagesh, Hunsur Nagendra; Singh, Manjeet; Sriram, Dharmarajan; Yogeeswari, Perumal; Sekhar, Kondapalli Venkata Gowri Chandra;
European Journal of Medicinal Chemistry, Year: 2015, Vol: 92, Pages: 415-426
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Synthesis and evaluation of 1-cyclopropyl-6-fluoro-1, 4-dihydro-4-oxo-7-(4-(2-(4-substitutedpiperazin-1-yl) acetyl) piperazin-1-yl) quinoline-3-carboxylic acid derivatives as anti-tubercular and antibacterial agents
Suresh, Narva; Nagesh, Hunsur Nagendra; Renuka, Janupally; Rajput, Vikrant; Sharma, Rashmi; Khan, Inshad Ali; Gowri, Chandra Sekhar Kondapalli Venkata;
European Journal of Medicinal Chemistry, Year: 2014, Vol: 71, Pages: 324-332
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Design, synthesis and antimycobacterial activity of various 3-(4-(substitutedsulfonyl) piperazin-1-yl) benzo [d] isoxazole derivatives
Naidu, Kalaga Mahalakshmi; Suresh, Amaroju; Subbalakshmi, Jayanty; Sriram, Dharmarajan; Yogeeswari, Perumal; Raghavaiah, Pallepogu; Sekhar, Kondapalli Venkata Gowri Chandra;
European Journal of Medicinal Chemistry, Year: 2014, Vol: 87, Pages: 71-78
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Design, synthesis and antimycobacterial evaluation of 1-(4-(2-substitutedthiazol-4-yl) phenethyl)-4-(3-(4-substitutedpiperazin-1-yl) alkyl) piperazine hybrid analogues
Nagesh, Hunsur Nagendra; Suresh, Amaroju; Sairam, Sirigina Devesh Sathya Sri; Sriram, Dharmarajan; Yogeeswari, Perumal; Sekhar, Kondapalli Venkata Gowri Chandra;
European Journal of Medicinal Chemistry, Year: 2014, Vol: 84, Pages: 605-613
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Synthesis and evaluation of anti-tubercular activity of 6-(4-substitutedpiperazin-1-yl) phenanthridine analogues
Nagesh, Hunsur Nagendra; Suresh, Narva; Naidu, Kalaga Mahalakshmi; Arun, Boyineni; Sridevi, Jonnalagadda Padma; Sriram, Dharmarajan; Yogeeswari, Perumal; Sekhar, Kondapalli Venkata Gowri Chandra;
European Journal of Medicinal Chemistry, Year: 2014, Vol: 74, Pages: 333-339
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Synthesis of novel ciprofloxacin analogues and evaluation of their anti-proliferative effect on human cancer cell lines
Suresh, Narva; Nagesh, Hunsur Nagendra; Sekhar, Kondapalli Venkata Gowri Chandra; Kumar, Anil; Shirazi, Amir N; Parang, Keykavous;
Bioorganic & medicinal chemistry letters, Year: 2013, Vol: 23, Pages: 6292-6295
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Design, synthesis, and preliminary in vitro and in vivo pharmacological evaluation of 4-{4-[2-(4-(2-substitutedquinoxalin-3-yl) piperazin-1-yl) ethyl] phenyl} thiazoles as atypical antipsychotic agents
Chandra Sekhar, Kondapalli Venkata Gowri; Rao, Vajja Sambasiva; Deuther-Conrad, Winnie; Sridhar, Divya; Nagesh, Hunsur Nagendra; Kumar, Vellas Sreedhar; Brust, Peter; Kumar, Muthyala Murali Krishna;
Medicinal Chemistry Research, Year: 2013, Vol: 22, Pages: 1660-1673
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Synthesis of 3, 5-diarylisoxazoles under solvent-free conditions using iodobenzene diacetate
Sekhar, Kondapalli Venkata Gowri Chandra; Sasank, Thripuraribhatla Venkata Naga Varuna Tara; Nagesh, Hunsur Nagendra; Suresh, Narva; Naidu, Kalaga Mahalakshmi; Suresh, Amaroju;
Chinese Chemical Letters, Year: 2013, Vol: 24, Pages: 1045-1048
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Design, synthesis and evaluation of 6-(4-((substituted-1H-1, 2, 3-triazol-4-yl) methyl) piperazin-1-yl) phenanthridine analogues as antimycobacterial agents
Nagesh, Hunsur Nagendra; Naidu, Kalaga Mahalakshmi; Rao, Damarla Harika; Sridevi, Jonnalagadda Padma; Sriram, Dharmarajan; Yogeeswari, Perumal; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic & Medicinal Chemistry Letters, Year: 2013, Vol: 23, Pages: 6805-6810
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Pharmacophore hypothesis for atypical antipsychotics
Sekhar, KVGC; Vyas, Devambhatla Ravi Kumar; Nagesh, Hunsur Nagendra; Rao, Vajja Sambasiva;
Bull. Korean Chem. Soc, Year: 2012, Vol: 33, Pages: 2930-2936
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Prevalence and risk factors of hypertension in above 40 years age group urban population of Kadapa
Chandra Sekhar, K; Moukthika, KVN; Krishna, C Bala; Kumar, KJ Kishore; Kumar, DS Sujith; Keshav, Suresh;
Public Health Research & Development, Year: 2011, Vol: 2, Pages: 30
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Synthesis of Triazoloquinoxalines as antitubercular agents
Sekhar, Kondapalli Venkata Gowri Chandra; Rao, Vajja Sambasiva; Kumar, Dalip;
Bulletin of the Korean Chemical Society, Year: 2011, Vol: 32, Pages: 2657-2660
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Design, synthesis, and preliminary in vitro and in vivo pharmacological evaluation of 2-{4-[4-(2, 5-disubstituted thiazol-4-yl) phenylethyl] piperazin-1-yl}-1, 8-naphthyridine-3-carbonitriles as atypical antipsychotic agents
Gowri Chandra Sekhar, Kondapalli Venkata; Rao, Vajja Samabasiva; Deuther-Conrad, Winnie; Reddy, Aravalli Satish; Brust, Peter; Krishna Kumar, Mutyala Murali;
Journal of Enzyme Inhibition and Medicinal Chemistry, Year: 2011, Vol: 26, Pages: 561-568
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Solvent free microwave accelerated synthesis of heterocyclic thiazolidin-4-ones as antimicrobial and antifungal agents
Sekhar, Kondapalli Venkata Gowri Chandra; Rao, Vajja Sambasiva; Reddy, Aravalli Satish; Sunandini, Ravada; Satuluri, VSA;
Bulletin of the Korean Chemical Society, Year: 2010, Vol: 31, Pages: 1219-1222
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Synthesis and preliminary screening of novel N-{2-[4-(substituted) piperazin-1-yl]-2-oxoethyl} acetamides as potential atypical antipsychotic agents
Chandra Sekhar, Kondapalli Venkata Gowri; Rao, Vajja Samabasiva; Krishna, Mutyala Murali;
Journal of Enzyme Inhibition and Medicinal Chemistry, Year: 2009, Vol: 24, Pages: 871-875
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Synthesis and Pharmacological Evaluation of Novel Heterocyclic Compounds as Potential Agents for the Treatment of Schizophrenia
KVG, Chandra Sekhar;
BITS PILANI, Year: 2008
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Synthesis and preliminary pharmacological evaluation of N-2-(4-(4-(2-substitutedthiazol-4-yl) piperazin-1-yl)-2-oxoethyl) acetamides as novel atypical antipsychotic agents
Sekhar, KVG Chandra; Rao, VS; Vyas, Devambatla Ravi Kumar; Kumar, M Murali Krishna;
Bioorganic & medicinal chemistry letters, Year: 2008, Vol: 18, Pages: 6054-6057
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Progress in the research of artemisinin and its analogues as antimalarials: an update
Sriram, Dharmarajan; Rao, Vajja Sambasiva; Chandrasekhar, Kondapalli Venkata Gowri; Yogeeswari, Perumal;
Natural Product Research, Year: 2004, Vol: 18, Pages: 503-527
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An expeditious synthesis of 1-aryl-4-methyl-1, 2, 4-triazolo [4, 3-a] quinoxalines under solvent-free conditions using iodobenzene diacetate
Kumar, Dalip; Chandra Sekhar, Kondapalli VG; Dhillon, Harmeet; Rao, Vajja S; Varma, Rajender S;
Green chemistry, Year: 2004, Vol: 6, Pages: 156-157
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Iodobenzene diacetate mediated solid?state synthesis of heterocyclyl?1, 3, 4?oxadiazoles
Rao, VS; Chandra Sekhar, KVG;
Synthetic communications, Year: 2004, Vol: 34, Pages: 2153-2157
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Determination of total arsenic concentration in clinical samples for epidemiological studies using ICP-MS
Chandra Sekhar, K; Chary, NS; Kamala, CT; Anupama, M; Reddy, MRP;
Atom. Spectros, Year: 2002, Vol: 23, Pages: 170-175
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Higher acyclic nitrogen containing deoxy sugar derivatives: a new lead in the generation of antimycobacterial chemotherapeutics
Pathak, Rashmi; Shaw, Arun K; Bhaduri, Amiya P; Chandrasekhar, KVG; Srivastava, Anil; Srivastava, Kishore K; Chaturvedi, Vineeta; Srivastava, Ranjana; Srivastava, Brahm S; Arora, Shalini;
Bioorganic & medicinal chemistry, Year: 2002, Vol: 10, Pages: 1695-1702