Professor Publications
One-Pot Diastereoselective Synthesis of Spiro [pyrimidine-5, 8?-thiazolo [5, 4-f] quinoline] triones and Diimidazo-pyrazinyl-bis (1, 3-dimethyl-2, 4, 6-trioxohexahydropyrimidine-5-ylium) dihydrate as Anticancer Agents
Parmar, Mehul P; Chaudhari, Hrushikesh S; Vala, Disha P; Macwan, Pradip M; Nogales, Joaquina; Sahoo, Subash C; Salunke, Deepak B; Banerjee, Sourav; Chandra Sekhar, Kondapalli Venkata Gowri; Khan, Adam N;
The Journal of Organic Chemistry
Discovery of triazole-tethered glycinate and propanoate derivatives bearing a thiolactone moiety as quorum sensing inhibitors of Pseudomonas aeruginosa: design, synthesis, biological evaluation, and biofilm inhibition
Chaitanya, Kosana Sai; Yu, Tsz Tin; Chaudhari, Hrushikesh; Orenkonday, Nidhi; Kuthe, Pranali Vijaykumar; Kumar, Naresh; Dey, Ruchi Jain; Murugesan, Sankaranarayanan; Gowri Chandra Sekhar, Kondapalli Venkata;
RSC advances, Vol. 16, No. 30, pp. 27977-27993
Nitro-thiochromene derivatives as promising anti-leishmanial agents: Synthesis, biological evaluation, and in silico insights
7. Jatin Malik, Estela Melcon-Fernandez, Rafael Balana Fouce, Chandra Sekhar Kondapalli Venkata Gowri, Murugesan Sankaranarayanan;
Journal of Molecular Structure, Vol. 1356, pp. 145170
Design, Synthesis and Evaluation of Indole?Based 1, 2, 3?Triazoles as Potential Quorum Sensing and Biofilm Inhibitors Against Pseudomonas aeruginosa
Chaitanya, Kosana Sai; Yu, Tsz Tin; Chaudhari, Hrushikesh; Orekonday, Nidhi; Kumar, Naresh; Dey, Ruchi Jain; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Archiv der Pharmazie, Vol. 359, No. 2, pp. e70209
Targeted HDAC8 inhibition with non-hydroxamate [1, 2, 4] triazolo [4, 3-a] quinoline compounds
Bandaru, NVM Rao; Fathima, Ashna; Sengar, Suryansh; Schweipert, Markus; Chaitanya, Kosana Sai; Mohammed, Muzaffar-Ur-Rehman; Gore, Suraj T; Jamma, Trinath; Sharma, Vivek; Abbineni, Chandrasekhar;
Scientific Reports, Vol. 16, No. 1, pp. 7472
Spirochromanone Cst-17 as a potent microtubule destabilizing agent showing anticancer effects in HeLa cells by binding to tubulin
5. Ranita Roy, Adinarayana Nandikolla, Debabrata Ghosh Dastidar, Urmi Chatterji, Kondapalli Venkata Gowri Chandra Sekhar, and Gopal Chakrabarti;
Scientific Publication
2-(1H-Pyrazol-1-yl) pyrimidine derivatives as promising anticancer candidates: synthesis, biological studies, and computational insights
Talamadla, Mahesh Kumar; Moharir, Shreyash Rajendra; Katdare, Mihika; Sengar, Suryansh; Sharma, Vivek; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Journal of Molecular Structure, pp. 145158
Recent advances in triazole hybrid molecules for the therapeutic management of neglected tropical diseases
Malik, Jatin; Karande, Gauri; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
RSC Medicinal Chemistry, Vol. 16, No. 11, pp. 5292-5317
Design, synthesis, and biological evaluation of (E)-3-amino-N?-substituted benzylidene-6-chloropyrazine-2-carbohydrazide derivatives as anti-mycobacterial agents
Kumar, Boddupalli Venkata Siva; Bhardwaj, Puja; Chaudhari, Hrushikesh S; Dey, Ruchi Jain; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic Chemistry, pp. 109206
Zinc based organic metal complexes for OLED applications
Paul, J John; Chaitanya, Kosana Sai; Ganesan, R; Jha, Purushottam; Sekhar, Kondapalli Venkata Gowri Chandra; Sindhu, S;
Synthetic Metals, pp. 117980
Harnessing SIRT1 activators for effective PCOS treatment: A new frontier
Moharir, Shreyash Rajendra; Talamadla, Mahesh Kumar; Bhardwaj, Puja; Banerjee, Arnab; Dey, Ruchi Jain; Sekhar, Kondapalli Venkata Gowri Chandra;
Biomedicine & Pharmacotherapy, Vol. 190, pp. 118361
Eco-friendly polyethylene glycol (PEG-400): PEG mediated synthesis, in-vitro, molecular dynamics, DFT, docking, ADMET and MM-GBSA studies of novel sulfonamides as potential antioxidant agents
Santhosh, CR; Chinnam, Sampath; Chaudhari, Hrushikesh S; Sekhar, Kondapalli Venkata Gowri Chandra; Oduselu, Gbolahan O; Ahuja, Vishal; Chidambaram, Kumarappan; Kerru, Nagaraju; Madhu, GM;
Journal of Molecular Structure, Vol. 1346, pp. 143201
Exploring the Anti?Tubercular Potential of 2?(1H?Pyrazol?1?yl) Pyrimidine: Design, Synthesis, Biological Evaluation and Molecular Docking Studies
Talamadla, Mahesh Kumar; Nandikolla, Adinarayana; Shobha, Singarapalle; Nayar, Pranav Pramod; Kumar, Muthyala Murali Krishna; Sankaranarayanan, Murugesan; Sekhar, Kondapalli Venkata Gowri Chandra;
Chemistry & Biodiversity, Vol. 22, No. 7, pp. e202500321
Exploration of quinoxaline triazoles as antimycobacterial agents: design, synthesis and biological evaluation
Kumar, Boddupalli Venkata Siva; Talamadla, Mahesh Kumar; Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Shetye, Gauri; Franzblau, Scott G; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic & Medicinal Chemistry Letters, Vol. 121, pp. 130177
A critique review of fetal hemoglobin modulators through targeting epigenetic regulators for the treatment of sickle cell disease
Ala, Chandu; Ramalingam, Sivaprakash; Gowri, Chandra Sekhar Kondapalli Venkata; Sankaranarayanan, Murugesan;
Life Sciences, Vol. 369, pp. 123536
Design, synthesis, and biological evaluation of substituted benzyl-triazolopyridine derivatives as non-hydroxamate based HDAC8 inhibitors
Bandaru, NVM Rao; Fathima, Ashna; Joshi, Vandana; Schweipert, Markus; Pathur, Obanna; Chaitanya, Kosana Sai; Jamma, Trinath; Sharma, Vivek; Abbineni, Chandrasekhar; Meyer-Almes, Franz-Josef;
European Journal of Medicinal Chemistry Reports, Vol. 13, pp. 100255
Design and Synthesis of Novel Spiro [Chromane?2, 4??Piperidin]?4?One Derivatives: Anti?Proliferative Investigation and Molecular Docking Studies
Nakka, Srinuvasu; Sengar, Suryansh; Sai Chaitanya, Kosana; Swati; Chandu, Ala; Sankaranarayanan, Murugesan; Sharma, Vivek; Devunuri, Nagaraju; Gowri Chandra Sekhar, Kondapalli Venkata;
Asian Journal of Organic Chemistry, Vol. 14, No. 2, pp. e202400604
Exploring 4-morpholinopyrrolo-[2, 3-d]-pyrimidine derivatives as novel anti-cancer agents: Design, synthesis and biological studies
Nakka, Srinuvasu; Chaitanya, Kosana Sai; Sengar, Suryansh; Chandu, Ala; Sankaranarayanan, Murugesan; Sharma, Vivek; Devunuri, Nagaraju; Sekhar, Kondapalli Venkata Gowri Chandra;
Journal of Molecular Structure, Vol. 1319, pp. 139565
Development and Biological Evaluation of Novel Spiro 4?Chromanones as Potent Quorum Sensing Inhibitors
Sai Chaitanya, Kosana; Gupta, Pooja; Chitti, Surendar; Khetmalis, Yogesh Mahadu; Chandu, Ala; Murugesan, Sankaranarayanan; Pasupuleti, Mukesh; Sekhar, Kondapalli Venkata Gowri Chandra;
Journal of Chemistry, Vol. 2024, No. 1, pp. 8227205
Design, synthesis, and anti-mycobacterial evaluation of 1, 8-naphthyridine-3-carbonitrile analogues
Khetmalis, Yogesh Mahadu; Shobha, Singarapalle; Nandikolla, Adinarayana; Chandu, Ala; Murugesan, Sankaranarayanan; Kumar, Muthyala Murali Krishna; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC advances, Vol. 14, No. 31, pp. 22676-22689
Recent developments in thiochromene chemistry
Murugappan, Solai; Kuthe, Pranali Vijaykumar; Sekhar, Kondapalli Venkata Gowri Chandra; Sankaranarayanan, Murugesan;
Organic & Biomolecular Chemistry, Vol. 22, No. 30, pp. 6045-6079
Design, synthesis and biological evaluation of novel pyrido-[2, 3-d]-pyrimidin-2-amine analogues as antimycobacterial agents
Kumar, Boddupalli Venkata Siva; Khetmalis, Yogesh Mahadu; Chaitanya, Kosana Sai; Chandu, Ala; Shetye, Gauri; Ma, Rui; Murugesan, Sankaranarayanan; Franzblau, Scott G; Sekhar, Kondapalli Venkata Gowri Chandra;
Journal of Molecular Structure, Vol. 1303, pp. 137600
Tetrahydroisoquinoline based 5-nitro-2-furoic acid derivatives: a promising new approach for anti-tubercular agents
Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Sangeetha, Guruvelli Padma Vijaya; Chandu, Ala; Swati; Kumar, Muthyala Murali Krishna; Sharma, Vivek; Murugesan, Sankaranarayanan; Chandra Sekhar, Kondapalli Venkata Gowri;
New Journal of Chemistry, Vol. 47, No. 32, pp. 15378-15389
Design, synthesis, and biological evaluation of novel quinazolin-4 (3H)-one-based histone deacetylase 6 (HDAC6) inhibitors for anticancer activity
Khetmalis, Yogesh Mahadu; Fathima, Ashna; Schweipert, Markus; Debarnot, C?cile; Bandaru, Naga Venkata Madhusudhan Rao; Murugesan, Sankaranarayanan; Jamma, Trinath; Meyer-Almes, Franz-Josef; Sekhar, Kondapalli Venkata Gowri Chandra;
International Journal of Molecular Sciences, Vol. 24, No. 13, pp. 11044
Design, synthesis and biological evaluation of phenanthridine amide and 1, 2, 3-triazole analogues against Mycobacterium tuberculosis
Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Venkata Siva Kumar, Boddupalli; Chandu, Ala; Karan Kumar, Banoth; Shetye, Gauri; Ma, Rui; Murugesan, Sankaranarayanan; Franzblau, Scott G; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC Medicinal Chemistry, Vol. 14, No. 8, pp. 1549-1561
Molecular-level strategic goals and repressors in Leishmaniasis?Integrated data to accelerate target-based heterocyclic scaffolds
Abirami, M; Kumar, Banoth Karan; Dey, Sanchita; Johri, Samridhi; Reguera, Rosa M; Bala?a-Fouce, Rafael; Sekhar, Kondapalli Venkata Gowri Chandra; Sankaranarayanan, Murugesan;
European Journal of Medicinal Chemistry, Vol. 257, pp. 115471
Visible light sensing of ions by a cyanoquinoxaline 1, 4-dioxide-based probe and its applications
Savita; Nandikolla, Adinarayana; Shukla, Adarash Kumar; Chandra Sekhar, Kondapalli Venkata Gowri; Bhattacharya, Anupam;
Dalton Transactions, Vol. 52, No. 13, pp. 4103-4111
Retrospective review of chromane analogues as anti-protozoal leads: a decade's worth of evolution
Jadhav, Snehal R; Karan Kumar, Banoth; Joshi, Renuka Parshuram; Suryakant, Chougule Kishor; Chandu, Ala; Muzaffar-Ur-Rehman, Mohammed; Khetmalis, Yogesh Mahadu; Nandikolla, Adinarayana; Murugesan, Sankaranarayan; Chandra Sekhar, Kondapalli VG;
Current Topics in Medicinal Chemistry, Vol. 23, No. 9, pp. 713-735
Design, synthesis, and antimycobacterial evaluation of novel tetrahydroisoquinoline hydrazide analogs
Kumar, Boddupalli Venkata Siva; Khetmalis, Yogesh Mahadu; Nandikolla, Adinarayana; Kumar, Banoth Karan; Van Calster, Kevin; Murugesan, Sankaranarayanan; Cappoen, Davie; Sekhar, Kondapalli Venkata Gowri Chandra;
Chemistry & Biodiversity, Vol. 20, No. 2, pp. e202200939
Design, synthesis, and biological evaluation of tetrahydroisoquinoline based hydroxamate derivatives as HDAC 6 inhibitors for cancer therapy
Khetmalis, Yogesh Mahadu; Shree, Bakhya; Kumar, Boddupalli Venkata Siva; Schweipert, Markus; Debarnot, C?cile; Ashna, Fathima; Sankaranarayanan, Murugesan; Trinath, Jamma; Sharma, Vivek; Meyer-Almes, Franz-Josef;
Journal of Molecular Structure, Vol. 1278, pp. 134952
Inspection of in-house designed novel thiochromone amino-acid conjugate derivatives as Lm-NMT inhibitor?An in-silico analysis
Johri, Samridhi; Kumar, Banoth Karan; Dey, Sanchita; Balana-Fouce, Rafael; Sekhar, Kondapalli Venkata Gowri Chandra; Kunjiappan, Selvaraj; Murugesan, Sankaranarayanan;
Journal of Molecular Graphics and Modelling, Vol. 119, pp. 108397
Design, Synthesis and Biological Evaluation of Novel Spiro?[Chroman?2, 4??Piperidin]?4?One Analogs as Anti?Tubercular Agents
Chitti, Surendar; Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Van Calster, Kevin; Kumar, Boddupalli Venkata Siva; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Cappoen, Davie; Sekhar, Kondapalli Venkata Gowri Chandra;
Chemistry & Biodiversity, Vol. 19, No. 8, pp. e202200304
Design, synthesis and biological evaluation of benzo-[d]-imidazo-[2, 1-b]-thiazole and imidazo-[2, 1-b]-thiazole carboxamide triazole derivatives as antimycobacterial agents
Chitti, Surendar; Van Calster, Kevin; Cappoen, Davie; Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Cos, Paul; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
RSC advances, Vol. 12, No. 35, pp. 22385-22401
Design, Synthesis and Anti-mycobacterial Evaluation of Imidazo-[1,2-a]-pyridine Analogues
Yogesh, M, K., Surendar, C., Anjani, U. W., Karan Kumar, B., Murali Krishna Kumar M., Murugesan, S., Chandra Sekhar, K.V.G;
RSC Medicinal Chemistry, Vol. 13, pp. 327-342
Discovery of potent antitubercular agents: Design, synthesis and biological evaluation of 4-(3-(4-substitutedpiperazin-1-yl)-quinoxalin-2-yl)-naphthalen-1-ol analogues
Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Naidu, Kalaga Mahalakshmi; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Toxicology in Vitro, Vol. 82, pp. 105370
Search for structurally diverse heterocyclic analogs as dual-acting antimalarial and antileishmanial agents: An overview
Dey, Sanchita; Johri, Samridhi; Abirami, M; Kumar, Banoth Karan; Taramelli, Donatella; Basilico, Nicoletta; Balana-Fouce, Rafael; Sekhar, Kondapalli Venkata Gowri Chandra; Murugesan, Sankaranarayanan;
European Journal of Medicinal Chemistry Reports, Vol. 4, pp. 100031
Design, synthesis and evaluation of novel ?-carboline ester analogues as potential anti-leishmanial agents
Karan Kumar, Banoth; Faheem; Balana Fouce, Rafael; Melcon-Fernandez, Estela; Perez-Pertejo Yolanda, Yolanda; Reguera, Rosa M; Adinarayana, Nandikolla; Chandra Sekhar, Kondapalli Venkata Gowri; Vanaparthi, Satheeshvarma; Murugesan, Sankaranarayan;
Journal of Biomolecular Structure and Dynamics, Vol. 40, No. 23, pp. 12592-12607
Liquid chromatography-mass spectrometric methods for trace quantification of potential genotoxic impurities in ivacaftor and lumacaftor
Panchakarla, RK; Ravi, PR; Mullangi, S; Kondapalli, VGCS;
Annales Pharmaceutiques Fran?aises, Vol. 80, No. 4, pp. 448-459
Design, synthesis, and biological evaluation of phenyl thiazole-based AR-V7 degraders
Bhumireddy, Archana; Bandaru, NVM Rao; Reddy, B Raghurami; Gore, Suraj T; Mukherjee, Subhendu; Balasubramanian, Wesley Roy; Kumar, V Sumanth; Alapati, Krishna Satya; Sekhar, Kondapalli Venkata Gowri Chandra; Nellore, Kavitha;
Bioorganic & Medicinal Chemistry Letters, Vol. 55, pp. 128448
Anti-infective potential of manzamine alkaloids-a review
Ashok, Penta; Kumar, Banoth K; Chander, Subhash; Chandra, Sekhar; Kondapalli, VG; Sankaranarayanan, Murugesan;
Medicinal Chemistry, Vol. 18, No. 6, pp. 629-654
Pharmacophore based virtual screening, molecular docking, molecular dynamics and MM-GBSA approach for identification of prospective SARS-CoV-2 inhibitor from natural product databases
Kumar, Banoth Karan; Faheem, n; Sekhar, Kondapalli Venkata Gowri Chandra; Ojha, Rupal; Prajapati, Vijay Kumar; Pai, Aravinda; Murugesan, Sankaranarayanan;
Journal of Biomolecular Structure and Dynamics, Vol. 40, No. 3, pp. 1363-1386
Medicinal chemistry perspectives of 1, 2, 3, 4-tetrahydroisoquinoline analogs?biological activities and SAR studies
Karan Kumar, Banoth; Sekhar, Chandra; Gowri, Kondapalli Venkata; Chander, Subhash; Kunjiappan, Selvaraj; Murugesan, Sankaranarayanan;
RSC advances, Vol. 11, No. 20, pp. 12254-12287
Selective and Sensitive UHPLC Method for the Trace Analysis of Formaldehyde in Drug Substance Using Fused-core Column Technology and Detailed Pre-column Derivatization study
Panchakarla, Ravi K; Ravi, Punna Rao; Chandra Sekhar, Kondapalli VG;
Current Pharmaceutical Analysis, Vol. 17, No. 2, pp. 201-209
Design, synthesis and evaluation of novel ?-carboline ester analogues as potential anti-leishmanial agents.
Banoth Karan Kumar, Faheem, Rafael Balana Fouce, Estela Melcon-Fernandez, Nandikolla Adinarayana, Kondapalli Venkata Gowri Chandra Sekhar, Satheeshvarma Vanaparthi & Sankaranarayan Murugesan;
Journal of Biomolecular Structure and Dynamics, pp. DOI: 10.1080/07391102.2021.1973564.
1,2,3,4-Tetrahydroisoquinoline (THIQ) as privileged scaffold for anticancer de novo drug design.
Faheem, Banoth Karan Kumar, Kondapalli Venkata Gowri Chandra Sekhar, Subhash Chander, Selvaraj Kunjiappan & Sankaranarayanan Murugesan;
Expert Opinion on Drug Discovery, Vol. 16, No. 10, pp. 1119-114
Liquid chromatography?tandem mass spectrometric method for trace quantification of ethyl methanesulfonate: a genotoxic impurity in dapoxetine hydrochloride
Ravi Kiran Panchakarla, Punna Rao Ravi, Kondapalli Venkata Gowri Chandra Sekhar;
Future Journal of Pharmaceutical Sciences, Vol. 7, pp. 91
1,8-naphthyridine derivatives: an updated review on recent advancements of their myriad biological activities.
Shivani Mithula, Adinarayana Nandikolla, Sankaranarayanan Murugesan & Venkata GCS Kondapalli;
Future Medicinal Chemistry, Vol. 13, No. 18, pp. 1591-1618
Novel phenanthridine amide analogs as potential anti-leishmanial agents: In vitro and in silico insights
Nandikolla, Adinarayana; Srinivasarao, Singireddi; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Aggarwal, Himanshu; Balana-Fouce, Rafael; Melc?n-Fernandez, Estela; P?rez-Pertejo, Yolanda; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic Chemistry, Vol. 117, pp. 105414
Oxindole and its derivatives: A review on recent progress in biological activities
Khetmalis, Yogesh Mahadu; Shivani, Mithula; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
Biomedicine & Pharmacotherapy, Vol. 141, pp. 111842
Design, synthesis and biological evaluation of 7?(5?((substituted?amino)-methyl)-thiophen?2?yl)-spiro-[chroman?2, 4??piperidin]?4?one hydrochloride analogues as anticancer agents
Chitti, Surendar; Pulya, Sravani; Nandikolla, Adinarayana; Patel, Tarun Kumar; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Ghosh, Balaram; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic Chemistry, Vol. 112, pp. 104865
Design, synthesis and biological evaluation of novel 1, 2, 3-triazole analogues of Imidazo-[1, 2-a]-pyridine-3-carboxamide against Mycobacterium tuberculosis
Nandikolla, Adinarayana; Srinivasarao, Singireddi; Khetmalis, Yogesh Mahadu; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Shetye, Gauri; Ma, Rui; Franzblau, Scott G; Sekhar, Kondapalli Venkata Gowri Chandra;
Toxicology in Vitro, Vol. 74, pp. 105137
Recent Update on the Anti-infective Potential of ?-carboline Analogs
Faheem; Kumar, Banoth K; Sekhar, Kondapalli Venkata GC; Kunjiappan, Selvaraj; Jamalis, Joazaizulfazli; Balana-Fouce, Rafael; Sankaranarayanan, Murugesan;
Mini reviews in medicinal chemistry, Vol. 21, No. 4, pp. 398-425
Seeking potent anti-tubercular agents: design and synthesis of substituted-N-(6-(4-(pyrazine-2-carbonyl) piperazine/homopiperazine-1-yl) pyridin-3-yl) benzamide derivatives as anti-tubercular agents (vol 10, pg 12272, 2020)
Srinivasarao, Singireddi; Nandikolla, Adinarayana; Suresh, Amaroju; Van Calster, Kevin; De Vooght, Linda; Cappoen, Davie; Ghosh, Balaram; Aggarwal, Himanshu; Murugesan, Sankaranarayanan; Sekhar, Kondapalli Venkata Gowri Chandra;
RSC ADVANCES, Vol. 10, No. 32, pp. 18907-18907
Synthesis, study of antileishmanial and antitrypanosomal activity of imidazo pyridine fused triazole analogues
Nandikolla, Adinarayana; Srinivasarao, Singireddi; Karan Kumar, Banoth; Murugesan, Sankaranarayanan; Aggarwal, Himanshu; Major, Louise L; Smith, Terry K; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC advances, Vol. 10, No. 63, pp. 38328-38343
Inhibitors of pantothenate synthetase of Mycobacterium tuberculosis?a medicinal chemist perspective
Suresh, Amaroju; Srinivasarao, Singireddi; Khetmalis, Yogesh Mahadu; Nizalapur, Shashidhar; Sankaranarayanan, Murugesan; Sekhar, Kondapalli Venkata Gowri Chandra;
RSC advances, Vol. 10, No. 61, pp. 37098-37115
Druggable targets of SARS-CoV-2 and treatment opportunities for COVID-19
Kumar, Banoth Karan; Sekhar, Kondapalli Venkata Gowri Chandra; Kunjiappan, Selvaraj; Jamalis, Joazaizulfazli; Bala?a-Fouce, Rafael; Tekwani, Babu L; Sankaranarayanan, Murugesan;
Bioorganic chemistry, Vol. 104, pp. 104269
Discovery of 1, 2, 3-triazole based quinoxaline-1, 4-di-N-oxide derivatives as potential anti-tubercular agents
Srinivasarao, Singireddi; Nandikolla, Adinarayana; Suresh, Amaroju; Ewa, Augustynowicz-Kopec; G?ogowska, Agnieszka; Ghosh, Balaram; Kumar, Banoth Karan; Murugesan, Sankaranarayanan; Pulya, Sravani; Aggarwal, Himanshu;
Bioorganic Chemistry, Vol. 100, pp. 103955
Seeking potent anti-tubercular agents: design and synthesis of substituted-N-(6-(4-(pyrazine-2-carbonyl) piperazine/homopiperazine-1-yl) pyridin-3-yl) benzamide derivatives as anti-tubercular agents
Srinivasarao, Singireddi; Nandikolla, Adinarayana; Suresh, Amaroju; Calster, Kevin Van; De Voogt, Linda; Cappoen, Davie; Ghosh, Balaram; Aggarwal, Himanshu; Murugesan, Sankaranarayanan; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC advances, Vol. 10, No. 21, pp. 12272-12288
Visible-Light-Mediated Tandem Sulfonylation/Cyclization of Vinyl Azides with Sulfonyl Hydrazines for the Synthesis of 6-(Sulfonylmethyl) phenanthridines under Mild Conditions
Mao, Liu-Liang; Quan, Li-Xia; Zhu, Xian-Hong; Ji, Cong-Bin; Zhou, An-Xi; Chen, Fayun; Zheng, Da-Gui;
Synlett, Vol. 30, No. 8, pp. 955-960
Design, synthesis and biological evaluation of 1, 2, 3-triazole based 2-aminobenzimidazoles as novel inhibitors of LasR dependent quorum sensing in Pseudomonas aeruginosa
Srinivasarao, Singireddi; Nandikolla, Adinarayana; Nizalapur, Shashidhar; Yu, Tsz Tin; Pulya, Sravani; Ghosh, Balaram; Murugesan, Sankaranarayanan; Kumar, Naresh; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC advances, Vol. 9, No. 50, pp. 29273-29292
Design, synthesis and biological evaluation of 2-(3, 4-dimethoxyphenyl)-6 (1, 2, 3, 6-tetrahydropyridin-4-yl) imidazo [1, 2-a] pyridine analogues as antiproliferative agents
Chitti, Surendar; Singireddi, SrinivasaRao; Reddy, Pochana Santosh Kumar; Trivedi, Prakruti; Bobde, Yamini; Kumar, Chandan; Rangan, Krishnan; Ghosh, Balaram; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic & Medicinal Chemistry Letters, Vol. 29, No. 18, pp. 2551-2558
Design, synthesis and anti-tumour activity of new pyrimidine-pyrrole appended triazoles
Thiriveedhi, Arunkumar; Nadh, Ratnakaram Venkata; Srinivasu, Navuluri; Bobde, Yamini; Ghosh, Balaram; Sekhar, Kondapalli Venkata Gowri Chandra;
Toxicology in Vitro, Vol. 60, pp. 87-96
Design, synthesis and biological evaluation of 5-(2-(4-(substituted benzo [d] isoxazol-3-yl) piperazin-1-yl) acetyl) indolin-2-one and 5-(2-(4-substitutedpiperazin-1-yl) acetyl) indolin-2-one analogues as novel anti-tubercular agents
Naidu, Kalaga Mahalakshmi; Gajanan, Rudresh Naik; Sekhar, Kondapalli Venkata Gowri Chandra;
Arabian Journal of Chemistry, Vol. 12, No. 8, pp. 2418-2429
Synthesis and activity of benzopiperidine, benzopyridine and phenyl piperazine based compounds against Leishmania infantum.
Subhash Chander, Subhash Chander; Penta Ashok, Penta Ashok; Reguera, RM; Perez-Pertejo, MY; Carbajo-Andres, R; Balana-Fouce, R; Sekhar, KVGC; Murugesan Sankaranarayanan, Murugesan Sankaranarayanan;
Scientific Publication
Experimental study of flow blurring twin fluid atomization concept using transparent injector
Murugan, R; Bollu, B; Sekhar, K; Kolhe, PS;
ICLASS 2018-14th International Conference on Liquid Atomization and Spray Systems, No. 160082
Sulfur?Assisted Deprotection of Methylene Nitrile Group: One?Pot Synthesis of 4?Substituted?2H?1, 2, 3?triazoles
Nagesh, Hunsur Nagendra; Singireddi, Srinivasarao; Suresh, Amaroju; Nizalapur, Shashidhar; Murugesan, Sankaranarayanan; Kanneboina, Kumar; Kumar, Naresh; Sekhar, Kondapalli Venkata Gowri Chandra;
ChemistrySelect, Vol. 3, No. 26, pp. 7565-7571
Synthesis and activity of benzopiperidine, benzopyridine and phenyl piperazine based compounds against Leishmania infantum
Chander, Subhash; Ashok, Penta; Reguera, Rosa M; Perez-Pertejo, M Yolanda; Carbajo-Andres, Ruben; Balana-Fouce, Rafael; Sekhar, Kondapalli Venkata Gowri Chandra; Sankaranarayanan, Murugesan;
Experimental parasitology, Vol. 189, pp. 49-60
Design, Synthesis and Biological Evaluation of Triazole?Containing 2?Phenylindole and Salicylic Acid as Quorum Sensing Inhibitors Against Pseudomonas aeruginosa
Srinivasarao, Singireddi; Nizalapur, Shashidhar; Yu, Tsz Tin; Wenholz, Daniel Stanley; Trivedi, Prakruti; Ghosh, Balaram; Rangan, Krishnan; Kumar, Naresh; Gowri Chandra Sekhar, Kondapalli Venkata;
ChemistrySelect, Vol. 3, No. 32, pp. 9170-9180
Anti-proliferative activity, molecular modeling studies and interaction with calf thymus DNA of novel ciprofloxacin analogues: NARVA SURESH et al
Suresh, Narva; Suresh, Amaroju; Yerramsetty, Suresh; Bhadra, Manika Pal; Alvala, Mallika; Sekhar, Kondapalli Venkata Gowri Chandra;
Journal of Chemical Sciences, Vol. 130, No. 9, pp. 121
Design, synthesis of 9H-fluorenone based 1,2,3-triazole analogues as Mycobacterium tuberculosis InhA inhibitors
Suresh, A., Srinivasarao, S., Agnieszka, Ewa, Mallika, A., Lherbet, C, Chandra Sekhar, K.V.G.;
Chemical biology and drug design, Vol. 91, pp. 1078-1086
Design and synthesis of 4-morpholino-6-(1, 2, 3, 6-tetrahydropyridin-4-yl)-N-(3, 4, 5-trimethoxyphenyl)-1, 3, 5-triazin-2-amine analogues as tubulin polymerization inhibitors
Narva, Suresh; Chitti, Surendar; Amaroju, Suresh; Bhattacharjee, Debanjan; Rao, Bala Bhaskara; Jain, Nishant; Alvala, Mallika; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic & Medicinal Chemistry Letters, Vol. 27, No. 16, pp. 3794-3801
Do spiroindolines have the potential to replace vesamicol as lead compound for the development of radioligands targeting the vesicular acetylcholine transporter?
Lindemann, Marcel; Deuther-Conrad, Winnie; Moldovan, Rares; Sekhar, Kondapalli Venkata Gowri Chandra; Brust, Peter; Wenzel, Barbara;
Bioorganic & Medicinal Chemistry, Vol. 25, No. 19, pp. 5107-5113
A Study on Socio Demographic Profile of Adult Female Smokers in Rural Areas of Srikakulam District, AP
Sravya, B; Susmitha, G; Chandra Sekhar, K; Mohan, Ch Rama; Deotale, PG;
Indian Journal of Public Health Research & Development, Vol. 7, No. 1
Synthesis and biological evaluation of pyrrolo [2, 3-b] pyridine analogues as antiproliferative agents and their interaction with calf thymus DNA
Narva, Suresh; Chitti, Surendar; Bala, Bhaskara Rao; Alvala, Mallika; Jain, Nishant; Kondapalli, Venkata Gowri Chandra Sekhar;
European Journal of Medicinal Chemistry, Vol. 114, pp. 220-231
Design, synthesis and biological evaluation of new substituted sulfonamide tetrazole derivatives as antitubercular agents
Suresh, Amaroju; Suresh, Narva; Misra, Sunil; Kumar, Muthyala Murali Krishna; Sekhar, Kondapalli Venkata Gowri Chandra;
ChemistrySelect, Vol. 1, No. 8, pp. 1705-1710
Multicomponent cascade reaction: dual role of copper in the synthesis of 1, 2, 3-triazole tethered benzimidazo [1, 2-a] quinoline and their photophysical studies
Nagesh, Hunsur Nagendra; Suresh, Amaroju; Reddy, Muthyala Nagarjuna; Suresh, Narva; Subbalakshmi, Jayanty; Chandra Sekhar, Kondapalli Venkata Gowri;
RSC advances, Vol. 6, No. 19, pp. 15884-15894
Seeking potent anti-tubercular agents: Design, synthesis, anti-tubercular activity and docking study of various ((triazoles/indole)-piperazin-1-yl/1, 4-diazepan-1-yl) benzo [d] isoxazole derivatives
Naidu, Kalaga Mahalakshmi; Srinivasarao, Singireddi; Agnieszka, Napi?rkowska; Ewa, Augustynowicz-Kope?; Kumar, Muthyala Murali Krishna; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic & medicinal chemistry letters, Vol. 26, No. 9, pp. 2245-2250
Identification and development of pyrazolo [4, 3-c] pyridine carboxamides as Mycobacterium tuberculosis pantothenate synthetase inhibitors
Amaroju, Suresh; Kalaga, Mahalakshmi Naidu; Srinivasarao, Singireddi; Napi?rkowska, Agnieszka; Augustynowicz-Kope?, Ewa; Murugesan, Sankaranarayanan; Chander, Subhash; Krishnan, Rangan; Chandra Sekhar, Kondapalli Venkata Gowri;
New Journal of Chemistry, Vol. 41, No. 1, pp. 347-357
A Study of Nutritional Status of Adolescent Girls of Social Welfare Hostels in and around Vijayawada City.
Shridevi, K; Nageshwara Rao, R; Madhavi, P; Chandra Sekhar, K; Deotale, PG;
Indian Journal of Public Health Research & Development, Vol. 6, No. 1
G, Biswas NN, Nizalapur S, Rice SA, Willcox M, Black DSt. C, Kumar N
Goh, WK; Gardner, CR; Chandra Sekhar, KV;
Bioorg. Med. Chem, Vol. 23, pp. 7366
Synthesis and biological evaluation of novel phenanthridinyl piperazine triazoles via click chemistry as anti-proliferative agents
Nagesh, Hunsur Nagendra; Suresh, Narva; Prakash, Gollapalli Venkata Subrahmanya Bhanu; Gupta, Samarth; Rao, Janapala Venkateswara; Sekhar, Kondapalli Venkata Gowri Chandra;
Medicinal Chemistry Research, Vol. 24, No. 2, pp. 523-532
Novel amide and sulphonamide derivatives of 6-(piperazin-1-yl) phenanthridine as potent Mycobacterium tuberculosis H37Rv inhibitors
Naidu, Kalaga Mahalakshmi; Nagesh, Hunsur Nagendra; Singh, Manjeet; Sriram, Dharmarajan; Yogeeswari, Perumal; Sekhar, Kondapalli Venkata Gowri Chandra;
European Journal of Medicinal Chemistry, Vol. 92, pp. 415-426
Synthesis and evaluation of 1-cyclopropyl-6-fluoro-1, 4-dihydro-4-oxo-7-(4-(2-(4-substitutedpiperazin-1-yl) acetyl) piperazin-1-yl) quinoline-3-carboxylic acid derivatives as anti-tubercular and antibacterial agents
Suresh, Narva; Nagesh, Hunsur Nagendra; Renuka, Janupally; Rajput, Vikrant; Sharma, Rashmi; Khan, Inshad Ali; Gowri, Chandra Sekhar Kondapalli Venkata;
European Journal of Medicinal Chemistry, Vol. 71, pp. 324-332
Design, synthesis and antimycobacterial activity of various 3-(4-(substitutedsulfonyl) piperazin-1-yl) benzo [d] isoxazole derivatives
Naidu, Kalaga Mahalakshmi; Suresh, Amaroju; Subbalakshmi, Jayanty; Sriram, Dharmarajan; Yogeeswari, Perumal; Raghavaiah, Pallepogu; Sekhar, Kondapalli Venkata Gowri Chandra;
European Journal of Medicinal Chemistry, Vol. 87, pp. 71-78
Design, synthesis and antimycobacterial evaluation of 1-(4-(2-substitutedthiazol-4-yl) phenethyl)-4-(3-(4-substitutedpiperazin-1-yl) alkyl) piperazine hybrid analogues
Nagesh, Hunsur Nagendra; Suresh, Amaroju; Sairam, Sirigina Devesh Sathya Sri; Sriram, Dharmarajan; Yogeeswari, Perumal; Sekhar, Kondapalli Venkata Gowri Chandra;
European Journal of Medicinal Chemistry, Vol. 84, pp. 605-613
Synthesis and evaluation of anti-tubercular activity of 6-(4-substitutedpiperazin-1-yl) phenanthridine analogues
Nagesh, Hunsur Nagendra; Suresh, Narva; Naidu, Kalaga Mahalakshmi; Arun, Boyineni; Sridevi, Jonnalagadda Padma; Sriram, Dharmarajan; Yogeeswari, Perumal; Sekhar, Kondapalli Venkata Gowri Chandra;
European Journal of Medicinal Chemistry, Vol. 74, pp. 333-339
Synthesis of novel ciprofloxacin analogues and evaluation of their anti-proliferative effect on human cancer cell lines
Suresh, Narva; Nagesh, Hunsur Nagendra; Sekhar, Kondapalli Venkata Gowri Chandra; Kumar, Anil; Shirazi, Amir N; Parang, Keykavous;
Bioorganic & medicinal chemistry letters, Vol. 23, No. 23, pp. 6292-6295
Design, synthesis, and preliminary in vitro and in vivo pharmacological evaluation of 4-{4-[2-(4-(2-substitutedquinoxalin-3-yl) piperazin-1-yl) ethyl] phenyl} thiazoles as atypical antipsychotic agents
Chandra Sekhar, Kondapalli Venkata Gowri; Rao, Vajja Sambasiva; Deuther-Conrad, Winnie; Sridhar, Divya; Nagesh, Hunsur Nagendra; Kumar, Vellas Sreedhar; Brust, Peter; Kumar, Muthyala Murali Krishna;
Medicinal Chemistry Research, Vol. 22, No. 4, pp. 1660-1673
Synthesis of 3, 5-diarylisoxazoles under solvent-free conditions using iodobenzene diacetate
Sekhar, Kondapalli Venkata Gowri Chandra; Sasank, Thripuraribhatla Venkata Naga Varuna Tara; Nagesh, Hunsur Nagendra; Suresh, Narva; Naidu, Kalaga Mahalakshmi; Suresh, Amaroju;
Chinese Chemical Letters, Vol. 24, No. 12, pp. 1045-1048
Design, synthesis and evaluation of 6-(4-((substituted-1H-1, 2, 3-triazol-4-yl) methyl) piperazin-1-yl) phenanthridine analogues as antimycobacterial agents
Nagesh, Hunsur Nagendra; Naidu, Kalaga Mahalakshmi; Rao, Damarla Harika; Sridevi, Jonnalagadda Padma; Sriram, Dharmarajan; Yogeeswari, Perumal; Sekhar, Kondapalli Venkata Gowri Chandra;
Bioorganic & Medicinal Chemistry Letters, Vol. 23, No. 24, pp. 6805-6810
Pharmacophore hypothesis for atypical antipsychotics
Sekhar, KVGC; Vyas, Devambhatla Ravi Kumar; Nagesh, Hunsur Nagendra; Rao, Vajja Sambasiva;
Bull. Korean Chem. Soc, Vol. 33, No. 9, pp. 2930-2936
Prevalence and risk factors of hypertension in above 40 years age group urban population of Kadapa
Chandra Sekhar, K; Moukthika, KVN; Krishna, C Bala; Kumar, KJ Kishore; Kumar, DS Sujith; Keshav, Suresh;
Public Health Research & Development, Vol. 2, No. 2, pp. 30
Synthesis of Triazoloquinoxalines as antitubercular agents
Sekhar, Kondapalli Venkata Gowri Chandra; Rao, Vajja Sambasiva; Kumar, Dalip;
Bulletin of the Korean Chemical Society, Vol. 32, No. 8, pp. 2657-2660
Design, synthesis, and preliminary in vitro and in vivo pharmacological evaluation of 2-{4-[4-(2, 5-disubstituted thiazol-4-yl) phenylethyl] piperazin-1-yl}-1, 8-naphthyridine-3-carbonitriles as atypical antipsychotic agents
Gowri Chandra Sekhar, Kondapalli Venkata; Rao, Vajja Samabasiva; Deuther-Conrad, Winnie; Reddy, Aravalli Satish; Brust, Peter; Krishna Kumar, Mutyala Murali;
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 26, No. 4, pp. 561-568
Solvent free microwave accelerated synthesis of heterocyclic thiazolidin-4-ones as antimicrobial and antifungal agents
Sekhar, Kondapalli Venkata Gowri Chandra; Rao, Vajja Sambasiva; Reddy, Aravalli Satish; Sunandini, Ravada; Satuluri, VSA;
Bulletin of the Korean Chemical Society, Vol. 31, No. 5, pp. 1219-1222
Synthesis and preliminary screening of novel N-{2-[4-(substituted) piperazin-1-yl]-2-oxoethyl} acetamides as potential atypical antipsychotic agents
Chandra Sekhar, Kondapalli Venkata Gowri; Rao, Vajja Samabasiva; Krishna, Mutyala Murali;
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 24, No. 3, pp. 871-875
Synthesis and Pharmacological Evaluation of Novel Heterocyclic Compounds as Potential Agents for the Treatment of Schizophrenia
KVG, Chandra Sekhar;
BITS PILANI
Synthesis and preliminary pharmacological evaluation of N-2-(4-(4-(2-substitutedthiazol-4-yl) piperazin-1-yl)-2-oxoethyl) acetamides as novel atypical antipsychotic agents
Sekhar, KVG Chandra; Rao, VS; Vyas, Devambatla Ravi Kumar; Kumar, M Murali Krishna;
Bioorganic & medicinal chemistry letters, Vol. 18, No. 23, pp. 6054-6057
Progress in the research of artemisinin and its analogues as antimalarials: an update
Sriram, Dharmarajan; Rao, Vajja Sambasiva; Chandrasekhar, Kondapalli Venkata Gowri; Yogeeswari, Perumal;
Natural Product Research, Vol. 18, No. 6, pp. 503-527
An expeditious synthesis of 1-aryl-4-methyl-1, 2, 4-triazolo [4, 3-a] quinoxalines under solvent-free conditions using iodobenzene diacetate
Kumar, Dalip; Chandra Sekhar, Kondapalli VG; Dhillon, Harmeet; Rao, Vajja S; Varma, Rajender S;
Green chemistry, Vol. 6, No. 3, pp. 156-157
Iodobenzene diacetate mediated solid?state synthesis of heterocyclyl?1, 3, 4?oxadiazoles
Rao, VS; Chandra Sekhar, KVG;
Synthetic communications, Vol. 34, No. 12, pp. 2153-2157
Determination of total arsenic concentration in clinical samples for epidemiological studies using ICP-MS
Chandra Sekhar, K; Chary, NS; Kamala, CT; Anupama, M; Reddy, MRP;
Atom. Spectros, Vol. 23, No. 5, pp. 170-175
Higher acyclic nitrogen containing deoxy sugar derivatives: a new lead in the generation of antimycobacterial chemotherapeutics
Pathak, Rashmi; Shaw, Arun K; Bhaduri, Amiya P; Chandrasekhar, KVG; Srivastava, Anil; Srivastava, Kishore K; Chaturvedi, Vineeta; Srivastava, Ranjana; Srivastava, Brahm S; Arora, Shalini;
Bioorganic & medicinal chemistry, Vol. 10, No. 6, pp. 1695-1702